Synthesis and antimicrobial activity of some novel heterocycles containing thiazole, oxazole, thiazine, oxazine and triazole moiety

Journal of the Iranian Chemical Research

مقاله 5، دوره 4، شماره 1، خرداد 2011، صفحه 33-38   

نویسندگان

Vijay V. Dabholkar^* ؛ Sunil R. Patil؛ Rajesh V. Pandey

Organic Research Laboratory, Department of Chemistry, KC College, Churchgate, Mumbai, India

چکیده

Indandione 1 was brominated to yield 2-bromoIndandione 2 which on further reacted with substituted thiocarbamides, carbamides, 2-aminothiophenols, 2-aminophenol and triazoles to furnished 3-substituted aniline-2-thia-4-aza-6,7-benzo-8-oxo-bicyclo [3.3.0]-1(5),3-octadiene 3, 3-substituted aniline-2-oxa-4-aza-6,7-benzo-8-oxo-bicyclo [3.3.0]-1(5),3-octadiene 4, 2-Thia-5-aza-9-oxo-3,4-(3’-substituted) benzo-7,8-benzo-bicyclo [4.3.0]-1(6) nonene 5, 2-oxa-5-aza-9-oxo-(3, 4)-(7, 8)-dibenzo-bicyclo [4.3.0]-1(6) nonene 6, 3-substituted-(1,2,4) triazolo [4,5-b] [indeno (2,3-e)]-1,3,4-thiadiazine 7 respectively.

کلیدواژه‌ها

Monobromoindandione؛ Thiocarbamide؛ Carbamide؛ 2-Aminothiophenol؛ 2-Aminophenol؛ triazole

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